PMID- 27267124
OWN - NLM
STAT- PubMed-not-MEDLINE
DCOM- 20180516
LR  - 20180516
IS  - 1520-6904 (Electronic)
IS  - 0022-3263 (Linking)
VI  - 81
IP  - 13
DP  - 2016 Jul 1
TI  - One-Pot Synthesis of Substituted Benzo[b]furans and Indoles from 
      Dichlorophenols/Dichloroanilines Using a Palladium-Dihydroxyterphenylphosphine 
      Catalyst.
PG  - 5450-63
LID - 10.1021/acs.joc.6b00824 [doi]
AB  - Disubstituted benzo[b]furans were synthesized by ortho-selective Sonogashira 
      coupling of dichlorophenols and terminal alkynes, followed by cyclization and 
      Suzuki-Miyaura coupling in one pot, using a palladium-dihydroxyterphenylphosphine 
      (Cy-DHTP) catalyst. The use of substoichiometric amounts of tetrabutylammonium 
      chloride was effective in accelerating the Suzuki-Miyaura coupling. This protocol 
      was also successfully applied to the one-pot synthesis of disubstituted indoles 
      from dichloroaniline derivatives.
FAU - Yamaguchi, Miyuki
AU  - Yamaguchi M
AD  - School of Pharmaceutical Sciences, University of Shizuoka , 52-1 Yada, Suruga-ku, 
      Shizuoka 422-8526, Japan.
FAU - Akiyama, Tomoyo
AU  - Akiyama T
AD  - School of Pharmaceutical Sciences, University of Shizuoka , 52-1 Yada, Suruga-ku, 
      Shizuoka 422-8526, Japan.
FAU - Sasou, Hirohisa
AU  - Sasou H
AD  - School of Pharmaceutical Sciences, University of Shizuoka , 52-1 Yada, Suruga-ku, 
      Shizuoka 422-8526, Japan.
FAU - Katsumata, Haruka
AU  - Katsumata H
AD  - School of Pharmaceutical Sciences, University of Shizuoka , 52-1 Yada, Suruga-ku, 
      Shizuoka 422-8526, Japan.
FAU - Manabe, Kei
AU  - Manabe K
AD  - School of Pharmaceutical Sciences, University of Shizuoka , 52-1 Yada, Suruga-ku, 
      Shizuoka 422-8526, Japan.
LA  - eng
PT  - Journal Article
PT  - Research Support, Non-U.S. Gov't
DEP - 20160614
PL  - United States
TA  - J Org Chem
JT  - The Journal of organic chemistry
JID - 2985193R
EDAT- 2016/06/09 06:00
MHDA- 2016/06/09 06:01
CRDT- 2016/06/09 06:00
PHST- 2016/06/09 06:00 [entrez]
PHST- 2016/06/09 06:00 [pubmed]
PHST- 2016/06/09 06:01 [medline]
AID - 10.1021/acs.joc.6b00824 [doi]
PST - ppublish
SO  - J Org Chem. 2016 Jul 1;81(13):5450-63. doi: 10.1021/acs.joc.6b00824. Epub 2016 
      Jun 14.